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Papers published by Professor Frank Boeckler:
Characterization of the Second-Generation Covalent Fragment Library (CovLib Gen2): Thiol Reactivity Profiling and p53-Y220C Rescue
Schwer M, Aldea SR, Engelhardt MU, Stahlecker J, Rheinganz J, Langkamp A, Boeckler FM
Drug Design, Development and Therapy 2026, 20:598622
Published Date: 18 May 2026
Standards for Computational Methods in Drug Design and Discovery: Simplified Guidance for Authors and Reviewers
Ibrahim TM, Hussain M, Boeckler FM
Drug Design, Development and Therapy 2025, 19:9649-9652
Published Date: 27 October 2025
Benchmarking the Structure-Based Virtual Screening Performance of Wild-Type and Resistant PfDHFR Using Docking and Machine Learning Re-Scoring
Hany MS, Ahmed NS, Boeckler FM, Ibrahim TM
Drug Design, Development and Therapy 2025, 19:7045-7058
Published Date: 15 August 2025
SNAr Reactive Pyrazine Derivatives as p53-Y220C Cleft Binders with Diverse Binding Modes
Klett T, Stahlecker J, Schwer M, Jaag SJ, Masberg B, Knappe C, Lämmerhofer M, Stehle T, Boeckler FM
Drug Design, Development and Therapy 2025, 19:4727-4753
Published Date: 3 June 2025
Screening of Covalent Kinase Inhibitors Yields Hits for Cysteine Protease USP7 / HAUSP
Ernst LN, Jaag SJ, Wydra VR, Masberg B, Knappe C, Gerstenecker S, Serafim RAM, Liang XJ, Seidler NJ, Lämmerhofer M, Gehringer M, Boeckler FM
Drug Design, Development and Therapy 2025, 19:2253-2284
Published Date: 25 March 2025
Evaluation of a Covalent Library of Diverse Warheads (CovLib) Binding to JNK3, USP7, or p53
Klett T, Schwer M, Ernst LN, Engelhardt MU, Jaag SJ, Masberg B, Knappe C, Lämmerhofer M, Gehringer M, Boeckler FM
Drug Design, Development and Therapy 2024, 18:2653-2679
Published Date: 1 July 2024
Statistical Analysis in Clinical and Experimental Medical Research: Simplified Guidance for Authors and Reviewers
Panos GD, Boeckler FM
Drug Design, Development and Therapy 2023, 17:1959-1961
Published Date: 3 July 2023
Synthesis of Amino Acids Bearing Halodifluoromethyl Moieties and Their Application to p53-Derived Peptides Binding to Mdm2/Mdm4
Vaas S, Zimmermann MO, Klett T, Boeckler FM
Drug Design, Development and Therapy 2023, 17:1247-1274
Published Date: 25 April 2023
Small-Molecule Intervention At The Dimerization Interface Of Survivin By Novel Rigidized Scaffolds
Ibrahim TM, Ernst C, Lange A, Hennig S, Boeckler FM
Drug Design, Development and Therapy 2019, 13:4247-4263
Published Date: 18 December 2019
Symmetric dimeric adamantanes for exploring the structure of two viroporins: influenza virus M2 and hepatitis C virus p7
Mandour YM, Breitinger U, Ma C, Wang J, Boeckler FM, Breitinger HG, Zlotos DP
Drug Design, Development and Therapy 2018, 12:1019-1031
Published Date: 30 April 2018