Back to User profile » Mr Jason Stahlecker

Papers published by Mr Jason Stahlecker:


Characterization of the Second-Generation Covalent Fragment Library (CovLib Gen2): Thiol Reactivity Profiling and p53-Y220C Rescue

Schwer M, Aldea SR, Engelhardt MU, Stahlecker J, Rheinganz J, Langkamp A, Boeckler FM

Drug Design, Development and Therapy 2026, 20:598622

Published Date: 18 May 2026

SNAr Reactive Pyrazine Derivatives as p53-Y220C Cleft Binders with Diverse Binding Modes

Graphical Abstract of SNAr Reactive Pyrazine Derivatives as p53-Y220C Cleft Binders with Diverse Binding Modes

Klett T, Stahlecker J, Schwer M, Jaag SJ, Masberg B, Knappe C, Lämmerhofer M, Stehle T, Boeckler FM

Drug Design, Development and Therapy 2025, 19:4727-4753

Published Date: 3 June 2025